TRPV3-74a

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TRPV3-74a
Identifiers
  • 3-[(S)-hydroxy(pyridin-2-yl)methyl]-1-methyl-3-[4-(trifluoromethyl)pyridin-2-yl]cyclobutan-1-ol
JSmol)
  • C[C@]1(C[C@@]([C@@H](C2=CC=CC=N2)O)(C3=CC(C(F)(F)F)=CC=N3)C1)O
  • InChI=1S/C17H17F3N2O2/c1-15(24)9-16(10-15,14(23)12-4-2-3-6-21-12)13-8-11(5-7-22-13)17(18,19)20/h2-8,14,23-24H,9-10H2,1H3/t14-,15?,16?/m1/s1
  • Key:MTJXDHFAWXGXIN-QQFBHYJXSA-N

TRPV3-74a is a drug which acts as a selective

antagonist for the TRPV3 calcium channel. It has analgesic effects in animal studies against both neuropathic pain and normal pain responses.[1][2]

References

  1. PMID 27077528
    .
  2. S2CID 100058677
    .


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