Atiprosin

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Atiprosin
Clinical data
Other namesAY-28,228
Routes of
administration		Oral
ATC code
  • none
Identifiers
  • (4aR,12bS)-1-ethyl-12-methyl-4-(propan-2-yl)-1,2,3,4,4a,5,6,12b-octahydropyrazino[2',3':3,4]pyrido[1,2-a]indole
JSmol)
  • n23c1ccccc1c(c2[C@H]4N(CCN([C@@H]4CC3)C(C)C)CC)C
  • InChI=1S/C20H29N3/c1-5-21-12-13-22(14(2)3)18-10-11-23-17-9-7-6-8-16(17)15(4)19(23)20(18)21/h6-9,14,18,20H,5,10-13H2,1-4H3/t18-,20+/m1/s1 checkY
  • Key:WXNVFYIBELASJW-QUCCMNQESA-N checkY
 ☒NcheckY (what is this?)  (verify)

Atiprosin (developmental code name AY-28,228) is an

antihypertensive agent which acts as a selective α1-adrenergic receptor antagonist.[1][2][3][4] It also possesses some antihistamine activity, though it is some 15-fold weaker in this regard than as an alpha blocker.[3] It was never marketed.[1]

See also

References

  1. ^
    ISBN 0-412-46630-9
    .
  2. PMID 3806618
    .
  3. ^
    S2CID 9361176
    .
  4. S2CID 19086175
    .

External links

  • Media related to Atiprosin at Wikimedia Commons
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