Epinastine

Source: Wikipedia, the free encyclopedia.
Epinastine
Clinical data
Trade namesAlesion, Elestat, Purivist, Relestat
AHFS/Drugs.comMonograph
MedlinePlusa604011
Pregnancy
category
  • C
Eye drops
ATC code
Pharmacokinetic data
Protein binding64%
Elimination half-life12 hours
Identifiers
  • (RS)-3-amino-9,13b-dihydro-1H-dibenz(c,f)imidazo(1,5-a)azepine
JSmol)
  • N\4=C(\N3c1c(cccc1)Cc2c(cccc2)C3C/4)N
  • InChI=1S/C16H15N3/c17-16-18-10-15-13-7-3-1-5-11(13)9-12-6-2-4-8-14(12)19(15)16/h1-8,15H,9-10H2,(H2,17,18) checkY
  • Key:WHWZLSFABNNENI-UHFFFAOYSA-N checkY
  (verify)

Epinastine (brand names Alesion, Elestat, Purivist, Relestat) is a second-generation

blood-brain-barrier.[2]

It was patented in 1980 and came into medical use in 1994.[3]

References