Bazinaprine

Source: Wikipedia, the free encyclopedia.
Bazinaprine
Clinical data
ATC code
  • None
Identifiers
  • 3-{[2-(morpholin-4-yl)ethyl]amino}-6-phenylpyridazine-4-carbonitrile
JSmol)
  • N#Cc2cc(nnc2NCCN1CCOCC1)c3ccccc3
  • InChI=1S/C17H19N5O/c18-13-15-12-16(14-4-2-1-3-5-14)20-21-17(15)19-6-7-22-8-10-23-11-9-22/h1-5,12H,6-11H2,(H,19,21) checkY
  • Key:KRNDIPHOJLIHRI-UHFFFAOYSA-N checkY
 ☒NcheckY (what is this?)  (verify)

Bazinaprine (SR-95,191) is an experimental drug candidate. It is a monoamine oxidase inhibitor (MAOI) which is believed to be useful for the treatment of depression. The drug strongly inhibits type A monoamine oxidase, but only weakly inhibits type B. The effects of the drug are reversible in vivo, but not in vitro.[1] In studies, the chemical has been shown to not interact in vivo with other neurotransmitter or drug receptor sites.[2]

See also

  • Reversible inhibitor of MAO-A
    (RIMA)

References