LS-115509

Add links
Source: Wikipedia, the free encyclopedia.
LS-115509
Clinical data
ATC code
  • none
Identifiers
  • 4-ethoxy-4-(furan-2-yl)-3-methyl-1-(2-phenylethyl)piperidine
JSmol)
  • CCOC1(CCN(CC1C)CCC2=CC=CC=C2)C3=CC=CO3
  • InChI=1S/C20H27NO2/c1-3-23-20(19-10-7-15-22-19)12-14-21(16-17(20)2)13-11-18-8-5-4-6-9-18/h4-10,15,17H,3,11-14,16H2,1-2H3
  • Key:INLMDDDTZIKNNI-UHFFFAOYSA-N

LS-115509 is an

4-phenylpiperidine family. It is comparable to drugs such as prodine and pheneridine, but is distinguished by the presence of an ether group and furan ring at the piperidine 4-position, which are not found in other drugs of this class. In animal studies, it has around 2-3x the potency of morphine depending on what assay is used. Like prodine, it has two stereocenters and four possible enantiomers, but the activity of these has not been tested separately.[1][2][3]

See also

References

  1. PMID 13877295
    .
  2. PMID 5319798
    .
  3. ISBN 978-0-12-443830-9
    .



Stub icon

This analgesic-related article is a stub. You can help Wikipedia by expanding it.

Retrieved from "https://en.wikipedia.org/w/index.php?title=LS-115509&oldid=1147962464"