Bezitramide

Source: Wikipedia, the free encyclopedia.
Bezitramide
Clinical data
Routes of
administration		Oral
ATC code
Legal status
Legal status
Identifiers
  • 4-[4-(2-oxo-3-propanoyl-2,3-dihydro-1H-benzimidazol-1-yl)piperidin-1-yl]-2,2-diphenylbutanenitrile
JSmol)
  • O=C(N2c1ccccc1N(C2=O)C5CCN(CCC(C#N)(c3ccccc3)c4ccccc4)CC5)CC
  • InChI=1S/C31H32N4O2/c1-2-29(36)35-28-16-10-9-15-27(28)34(30(35)37)26-17-20-33(21-18-26)22-19-31(23-32,24-11-5-3-6-12-24)25-13-7-4-8-14-25/h3-16,26H,2,17-22H2,1H3 checkY
  • Key:FLKWNFFCSSJANB-UHFFFAOYSA-N checkY
  (verify)

Bezitramide is an opioid

Janssen Pharmaceutica in 1961.[3][4][5]
It is most commonly marketed under the trade name Burgodin.

The drug was pulled from the shelves in the Netherlands in 2004 after fatal overdose cases, including one where a five-year-old child took one tablet from his mother's purse, ate it, and promptly died.[6]

Bezitramide is regulated much the same as morphine in all known jurisdictions and is a Schedule II substance under the United States' Controlled Substances Act of 1970, with an ACSCN of 9800 and zero annual manufacturing quota.[7] However, as of May 2021, it has never been marketed in the United States.

See also

References

  1. ^ Anvisa (2023-03-31). "RDC Nº 784 - Listas de Substâncias Entorpecentes, Psicotrópicas, Precursoras e Outras sob Controle Especial" [Collegiate Board Resolution No. 784 - Lists of Narcotic, Psychotropic, Precursor, and Other Substances under Special Control] (in Brazilian Portuguese). Diário Oficial da União (published 2023-04-04). Archived from the original on 2023-08-03. Retrieved 2023-08-16.
  2. S2CID 23978449
    .
  3. ^ US patent 3196157, Janssen PA, "Benzimidalinyl Piperidines", published 1963-06-11, issued 1965-07-20 
  4. PMID 5109278
    .
  5. PMID 4913411
    .
  6. PMID 6633692
    .
  7. ^ "Title 21 United States Code (USC) Controlled Substances Act". Archived from the original on 2020-08-30. Retrieved 2011-09-29.


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